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Ainm toraidh |
Gs441524 |
Coltas |
Pùdar geal, pill, seòrsa leaghan |
Assay |
> 99% |
Deuchainn |
HPLC |
CAS |
1191237-69-0 |
MF |
C12H13N5O4 |
Teòthachd stòraidh |
Àite tioram fionnar |
Ro-ràdh
Tha GS-441524 na phàirt gnìomhach bith-eòlasach de Remdesivir agus chaidh a chleachdadh gu farsaing air feadh an t-saoghail gus cait de peritonitis gabhaltach feline (FlP) a leigheas gu sàbhailte agus gu h-èifeachdach airson còrr air 18 mìosan. Tha FIP na ghalar cumanta agus gu math marbhtach ann an cait.
Gnìomh
Tha GS-441524 na mholacile beag le ainm saidheansail de inhibitor farpaiseach nucleoside triphosphate, a tha a ’nochdadh gnìomhachd anti-bhìoras làidir an aghaidh mòran bhìorasan RNA. Bidh e na substrate eile agus inneal-crìochnachaidh slabhraidh RNA airson RNA polymerase viral a tha an urra ri RNA. Tha an dùmhlachd neo-phuinnseanta de GS-441524 ann an ceallan feline cho àrd ri 100, a tha gu h-èifeachdach a’ bacadh ath-riochdachadh FIPV ann an cultar cealla CRFK agus macrophages peritoneal cat le galair nàdarra le dùmhlachd cho ìosal ri 1.
C: Dè a th' ann an GS?
A: Tha GS goirid airson GS-441524 a tha na dhroga anti-bhìorasach deuchainneach (nucleoside analog) a tha air cait a leigheas le FIP ann an deuchainnean achaidh a chaidh a dhèanamh aig UC Davis ach an Dr Neils Pedersen agus an sgioba aige. Faic sgrùdadh an seo.
Tha e an-dràsta ri fhaighinn mar in-stealladh no cungaidh-leigheis beòil ged nach eil an dreach beòil ri fhaighinn fhathast gu farsaing. Feuch an iarr thu air rianaire!
C: Dè cho fada 'sa tha an làimhseachadh?
F: Is e làimhseachadh a thathar a’ moladh stèidhichte air deuchainn làraich tùsail an Dotair Pedersen co-dhiù 12 seachdainean de in-stealladh fo-ghearradh làitheil.
Bu chòir obair-fala a sgrùdadh aig deireadh 12 seachdainean agus bu chòir comharran cait a mheasadh gus faicinn a bheil feum air làimhseachadh a bharrachd.
C: Dè dìreach a th’ ann an cùisean “neuro” no “ocular”?
A: Tha cat “Neuro” a’ ciallachadh gu bheil FIP air a dhol thairis air cnap-starra eanchainn fala agus tha comharraidhean a’ toirt a-steach cùisean siostam nearbhach meadhanach. Ataxia (laigse nam chasan cùil gu sònraichte), neo-chomas leum gu h-iomlan gun leisg, dìth co-òrdanachaidh agus faodaidh glacaidhean tachairt. Tha com-pàirt sùla, a tha cumanta leis an fhoirm eanchainn leis gu bheil na sùilean agus an eanchainn ceangailte gu dlùth, a’ coimhead mar seo:
C: Ciamar a bheir mi na stealladh GS?
A: Tha na stealladh air an toirt seachad fo-ghearradh no “fo-cu” a tha a’ ciallachadh dìreach fon chraiceann. Feumar in-stealladh a thoirt seachad a h-uile 24 uair cho faisg air an aon àm a h-uile latha sa ghabhas airson co-dhiù 12 seachdainean. CHAN EIL an t-snàthad a’ dol a-steach do fhèith a’ chait. Bidh an GS a’ stad air an in-stealladh ach tha am pian seachad cho luath ‘s a bhios an in-stealladh seachad. Tha grunn bhideothan cuideachail ann a tha na buill againn air post a chuir a’ sealltainn mar a bhios iad a’ stealladh agus cuideachd mòran air YouTube. Tha e nas fheàrr do lighiche-sprèidh a’ chiad in-stealladh no dhà a dhèanamh agus do theagasg mar a nì thu iad. Is dòcha gum feum piseagan a tha nas duilghe stad a chuir orra airson na seallaidhean turasan làitheil chun lighiche-sprèidh
Pacadh:
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PS: tha sinn a 'gabhail ri gnàthachadh pacaidh.
Luingearachd:
Bidh sinn a’ cur bathar tro DHL, Fedex, UPS, TNT, post Sìona, NL Post agus teachdairean eile, cuideam bho 10g gu 1000kg no eadhon bulker.
Thèid mion-fhiosrachadh luingeis & sgrìobhainnean luingeis a thoirt seachad agus a chuir gu luchd-ceannach fhad ‘s a tha e deiseil.
Bidh sinn a’ cumail sùil air an luchd gus am faigh luchd-cleachdaidh fàilte mhath.
Às deidh bliadhnaichean de eòlas luingeis às-mhalairt, le luchd-cur air adhart proifeasanta agus eòlach, bidh sinn a’ dèanamh cinnteach gun tèid bathar a lìbhrigeadh ann an grunn dhòighean sàbhailte agus èifeachdach.
1kg/foil bag, 25kg/bag or drum (PV bag for inner packing, and aluminium foil bag for outer packing.)
20 tons/20ft container,
25 tons/40ft container,
Or follow the client's requirements.
Delivery : We have special line transportation, or we can give it to yourforwarder Our special line transport is to ensure safe delivery to yourdesignated location, can be free of customs clearance (FedEx /EMS UPSDHL/TNT)
Payment: t/t, paypal, alibaba trade assurance,western union,bitcoin...Allmeans are acceptable as long as they are convenient for you(We do not acceptL/C and D/P during coronavirus)
Package:To better ensure thesafety of your goods, professionalenvironmentally friendly, convenient and efficient packaging services will beprovided.(1kg/25kgs/160kgs/200kgs)
Hebei Weimiao Import and Export Trade Co., Ltd.is specialized inR&D, manufacturingand marketing APIS,pharmaceuticalintermediates, we have two affiliated manufacturers. More than 70percent products are exported to Europe,America, Japan and Southeast Asia.Our factory located in Hebei, a beautiful coastal cityin the east region of China.
In the pastt years,Hebei Weimiao Import and Export Trade Co., Ltd.has established its professional team and advanced managements.excels in product sourcing and customized products. Development ofnew fine chemical, custom synthesis has been a significant part ofour chemical's production.
With our policy:"Credibility, Quality and Customer First".Wesincerely wish to tightly cooperate with the clients who areinterested in our products.
1.High quality with competitive price.
2.All purity>99%.
3.We are manufacturer and can provide high quality products with factory price.
PRE-SALES
1.reply timely We supply from stock and can deliver the goods to youin time
2.visit factory We can show you around our production plant
3.sample service You can get a sample of the product you want to buy
AFTER-SALES
1.safety delivery If there is any problem in transit, our company willmake up for it
2.quality assurance We can provide you with the test report of theproduct
OUR SUPERIORITY
High quality product
Competitive price
Professional technical team
Good after-sales service
Mature transportation Experience