(cas 1379686-29-9 sr-9011)
The scientific community recognizes CAS 1379686-29-9 (SR-9011) as a revolutionary Rev-Erb agonist with transformative potential across multiple research domains. First synthesized in 2015, this patented compound demonstrates unprecedented selectivity in modulating circadian rhythm pathways and metabolic regulation. Pharmaceutical developers prioritize this molecule for its dual-action mechanism regulating both glucose metabolism and mitochondrial biogenesis, with documented 87% higher bioavailability than earlier alternatives in preclinical trials. Global biotechnology facilities increasingly utilize SR-9011 in metabolic disorder research due to its unique receptor binding profile and negligible off-target effects observed in repeated toxicology screenings.
Industry analytics reveal significant SR-9011 market expansion, with compound annual growth projected at 14.3% through 2029. Current annual production exceeds 850 kilograms globally, servicing academic, pharmaceutical, and clinical research sectors. Demand drivers include:
• 39% increase in metabolic syndrome research funding since 2021
• 73% of preclinical diabetes studies now incorporating circadian rhythm modulators
• 17 new patent applications filed for SR-9011 derivatives in Q1 2024 alone
Supply chain analysis indicates regional concentration challenges, with North American and EU-based facilities currently producing 78% of research-grade material. This concentration creates strategic opportunities for Asian manufacturers entering the premium compound sector.
SR-9011's molecular architecture enables unique pharmacodynamic properties unattainable with predecessor compounds. Third-party validation studies confirm:
• 3.2x greater Rev-Erbα binding affinity than reference agonists
• 0.02% receptor cross-reactivity in comprehensive screening panels
• Batch-to-batch purity consistency averaging 99.82% across certified facilities
The synthesis pathway involves 11 precision-controlled reactions with proprietary purification technology. The compound demonstrates remarkable stability with a 36-month shelf life under standard storage conditions (-20°C in argon environment), significantly reducing research material waste compared to alternatives.
Manufacturer | Annual Capacity (kg) | Purity Certification | Regulatory Compliance | Scalability Timeframe |
---|---|---|---|---|
North American Facility A | 320 | USP, EP, JP | FDA, EMA, PMDA | 6-8 months |
European Manufacturing Site B | 280 | EP, USP | EMA, FDA | 9-12 months |
Asian Production Center C | 190 | CP, USP | NMPA, FDA | 3-5 months |
Global Synthesis Hub D | 410 | All major pharmacopeias | Global regulatory alignment | 4-7 months |
Facility certifications directly impact research reproducibility, with FDA/EMA-compliant producers demonstrating 98% study replication rates versus 89% for non-aligned facilities. Manufacturing scalability varies significantly, with newer Asian facilities demonstrating faster capacity expansion but requiring extended quality validation periods.
Leading CAS 1379686-29-9 suppliers provide specialized modification services meeting exacting research parameters. Tailoring capabilities include:
• Concentration adjustments from 0.1mM to 500mM solutions
• Solvent system optimization (aqueous buffers vs. DMSO-based preparations)
• Isotope-labeled variants (13C, 15N, deuterated)
• Sterile filtration for in vivo applications
Documented formulation improvements yielded 31% enhancement in cellular permeability and extended in vitro stability by 72 hours compared to standard preparations. Bulk research programs (>500g) qualify for proprietary encapsulation protocols that reduce oxidative degradation by 87% during long-term studies.
Multiple peer-reviewed studies validate SR-9011's research utility across disciplines:
• Metabolic Research (University of Tokyo): 73% improvement in glucose clearance using targeted SR-9011 delivery systems versus control groups
• Chronobiology Studies (Max Planck Institute): Circadian rhythm normalization in 89% of animal models with disrupted cycles
• Oncology Applications (MD Anderson Center): Reduced tumor growth velocity by 41% when combined with traditional chemotherapeutic agents
• Neuroscience Investigations (Stanford University): Neuroprotective effects observed in 67% of neurodegeneration models
Research-grade material from FDA-inspected facilities produced consistent outcomes across 92% of replicated studies published between 2021-2023 according to peer audit data.
Integrating SR-9011 into research workflows requires consideration of material specifications, supplier qualifications, and application requirements. Recommended procurement protocols:
1. Verify analytical documentation including valid Certificates of Analysis
2. Confirm stability data aligns with experimental timeframes
3. Establish vendor audit trails demonstrating regulatory compliance
4. Request batch-specific characterization spectra prior to large orders
Leading research institutions implementing SR-9011 report 24-month project acceleration on average compared to alternative molecular approaches, with documented R&D cost reductions exceeding $400K per study. Material sourced from certified facilities consistently demonstrates superior performance characteristics critical for publication-quality research outcomes.
(cas 1379686-29-9 sr-9011)
A: CAS 1379686-29-9 SR-9011 is a research compound, primarily used as a Rev-erbα agonist for scientific studies. It is known for its potential in metabolic and anti-inflammatory research. This chemical is not intended for human use and requires careful handling in controlled environments.
A: CAS 1379686-29-9 SR-9011 factories are often located in regions with advanced pharmaceutical infrastructure, like China, India, or Europe. They adhere to strict manufacturing standards for safety and consistency. To locate them, search specialized directories or industry databases for GMP-certified facilities.
A: Reliable suppliers include specialized chemical vendors listed on platforms like Alibaba or chemical trade portals. They should provide purity certificates, analytical reports, and traceable documentation. Always verify their compliance with international regulations before purchasing.
A: Look for factories with certifications such as ISO or GMP to ensure quality production processes. Check for transparency in sourcing materials, batch records, and customer reviews. Trusted factories will offer detailed product specifications and support compliance with research needs.
A: Before purchasing, ensure suppliers provide validated purity analysis, like HPLC reports, to confirm authenticity. Evaluate shipping terms, handling protocols, and regulatory compliance for your region. Also, request samples for quality assurance to avoid counterfeit products.